General Information of Drug Metabolite (DM) (ID: DM003374)
DM Name
AG-1549 Metabolite C26
Full List of Drug-Metabolizing Enzyme (DME) Related to This DM
DME(s) Producing This DM through Metabolism
DME Name DME ID Reactant Reaction Related Drug REF
Cytochrome P450 3A1 (Cyp3a1) DMEN096 Oxidation - Oxidationn AG-1549 [1]
Cytochrome P450 3A2 (Cyp3a2) DMEN097 Oxidation - Oxidationn AG-1549 [1]
Full List of Drug(s) That Produce This DM By Metabolism
AG-1549 DR0267 Phase 1 Human immunodeficiency virus infection
References
1 Evaluation of capravirine as a CYP3A probe substrate: in vitro and in vivo metabolism of capravirine in rats and dogs

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